Hāʻawi ʻo AASraw i nā ʻano o ka pauka pohō kaumaha me ka lako paʻa, pau nā hana āpau ma lalo o ke kānāwai cGMP a hiki ke nānā ʻia ka maikaʻi i kēlā me kēia manawa. Eia kekahi, hiki ke kākoʻo ʻia ke kauoha nui me ka uku hoʻokūkū.
E kūʻai i ka pauda hoʻemi kaumaha
1. Weight Loss Drug History
ʻO nā kinona mua o nā mea kaulike, i kapaʻia he mau mea'āpana momona i kēlā manawa, i loaʻa i ka pauʻana o 1800s. ʻOiaiʻo ka lāʻau lapaʻau i hana i kekahi hopena koʻikoʻi nui, ua hoʻomauʻia ka hoʻohanaʻiaʻana a hiki i nā 1960s.
Ua hoʻokomoʻia kekahi lāʻau hou i kapaʻiaʻo Dinitrophenol i nā 1930s a ua lilo i mea kaulana loa i ka mālamaʻana i ka poho kaumaha. ʻO ka lāʻau lapaʻau kahi i hoʻoikaikaʻia i loko o ke kino, kōkua i ka pohō kaumaha.
Ma waena o ka 1950s, loaʻa nā amphetamines a lilo i mea lapaʻau maʻamau. Hoʻomaopopoʻo ia i nā lilo o nā kaumaha ma kaʻokiʻana i kaʻai. I loko o ke kaumaha, ua hoʻonuiʻia ka hopena o ka hanuʻana o ka pulmonary, a ka hopena o ka weheʻana mai ka mākete ma 1968.
Ma nā 1970s, ua lilo ka ephedrine i mea mālamaʻia no ke kaumaha o ke kaumaha. ʻO ka lāʻau lapaʻau, akā naʻe, ua hopena i kekahi mau meaʻino i hiki ai ke haʻiʻia he mea weliweli.
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2. Weight Loss Drug Classification
Hoʻopiliʻia nā lāʻau lapaʻau maʻamau iʻekolu mahele nui e like me kā lākou hana hana a penei:
(1) Hoʻopale i ka'āpana (Diet)
ʻO nā lāʻauʻona e hoʻohaʻahaʻa i kaʻai ka mea i kapaʻia he sympathomimetic agents. Hoʻomaʻa pinepine lākou i ka meaʻai i ka hoʻonāukiukiʻana i ka noho maʻalahi ma mua o ka mea maʻamau. ʻO kaʻoluʻolu ka "piha" a me ka loaʻaʻana o kaʻai. Hanaʻia nā mea e hoʻopili ai i ka mea hoʻohana i ka neurotransmitter i loko o ka lolo kanaka e hoʻomalu i ka'ōpū, i kapaʻiaʻo noradrenaline (NA).
Hoʻokaʻawale kēia mau lāʻau lapaʻau i kahi ʻano kemika like me NA a hiki; ʻO ka hopena e hoʻopaʻa i nā mea loaʻa like me ka noradrenaline. ʻO nā lāʻau lapaʻau hoʻi e hoʻomaikaʻi i ka hana noradrenaline i ka "waena hānai" o ka lolo kanaka, ka hypothalamus. ʻO ka hypothalamus kanaka ke hoʻomalu i ke koena o ka ikehu i loko o ke kino. Hoʻopili ʻia ka ʻike e pili ana i nā hale kūʻai ikehu pākahi i loko o ka hypothalamus e hoʻoponopono ai i ka ʻai a me ka makemake. ʻO ka hoʻopaʻa ʻana o Noradrenaline a me ka hana i loko o ka hypothalamus he hopena hōʻemi i ka ʻai. ʻO ia mau lāʻau lapaʻau penei:
❶ Lorcaserin HCL(Belviq) CAS: 1431697-94-7
❷ Rimonabant HCL CAS: 158681-13-1
❸ DNP CAS: 119-26-6
(2) Ka momona
Hiki i nā lāʻau lapaʻau ke hoʻopau i ka momona ke kōkua i ka lilo ʻana o ka momona ma o ka hoʻohaʻahaʻa ʻana i ka makemake, hoʻomaikaʻi i ka metabolism, a me ka mālama ʻana i ka ʻai olakino. Hiki iā lākou ke hoʻonui i ka hiki ke hoʻomaʻamaʻa ma o ka hoʻonui ʻana i ka ikehu a me ka nānā ʻana. ʻO ia mau lāʻau lapaʻau e like me:
❶ Synephrine CAS: 94-07-5
❷ DMAA/1,3-Dimethylpentylamine CAS: 13803-74-2
(3) Hoʻonui i ka digestion
ʻO kēia mau lāʻau lapaʻau kūpono e hana ai ma ka paleʻana me ka hikiʻana o ka'ōnaehana hōʻona e hoʻomohu i nā meaʻai e pono ai i ka meaʻai. No ka laʻana, uaʻikeʻiaʻo Orlistat e kāohi i ka momona o ka momona a no laila ke pale nei i ka hoʻonaninalu momona. Ua hoʻohanaʻia kekahi mau mea'ē aʻe i ka hoʻohaʻahaʻaʻana i ka caloric a me ka hōʻinoʻana i ka hōʻomi. Ma kēia pāhana, e kūkākūkā kākou i nā mea hou e pili ana i kēia mau lāʻau lapaʻau:
❶ Orlistat CAS: 96829-58-2
❷ Cetilistat CAS: 282526-98-1
3. ʻO 3 Loaʻa kaulana loa i ka pauda kaumaha ma ka mākeke
(1) Orlistat CAS: 96829-58-2
ʻO Orlistat kekahi mea hoʻokipa pāʻani pancreatic a me ka lipase lipid. Hoʻopiliʻia nā'āpana triglycerides a pau me ke kōkuaʻana o nā pancreatic and lipst lipases. Hiki i nā lipases enzymatically e hoʻohiolo i nā triglycerides i loko o nā mea momona momona liʻiliʻi e hiki ke hoʻomohuʻia ma hope o nā'ōpū liʻiliʻi. Hoʻopiliʻia nā mea pāpālua a me nā'āpana lipase Gastric a me ka pancreatic me nā pancreatic and lipstases i loko o ka lumen o ka'ōpū liʻiliʻi a me ka'ōpū e hana ana i kēia mau enzymes hikiʻole ke hana pono.
Ma o ka hanaʻoleʻana i nā hana o kēia mau lipases, hiki keʻaʻaʻia ka momona momona o nā meaʻai, a ua hoʻokuʻuʻia nā triglycerides i loko o nā feces. ʻO Orlistat ka lāʻau lapaʻau palekana e pale ai i ka 30 ka nui o nā momonaʻai mai kaʻaiʻana mai ka hoʻokomoʻana i ka'ōnaehana kino kanaka (i ka manawa o 30 ka nui o ka ikehu i nā meaʻai e nā triglycerides). ʻO ka emiʻana o ka haʻawina kaumaha ma hope o hoʻokahi makahiki me ka hui pūʻia o Xenical (orlistat) a me ka hoʻololiʻana i keʻano o ka nohoʻana, e puni ana i ka 8.5 kg.
Me ka laweʻana i ka laweʻana o nā triglycerides meaʻai, a iʻole e huli i ka paukū pau o nā meaʻai i:
- Loaʻa ka hopena maikaʻi i ke koko;
- E ho'ēmi i ka cholesterol absorption a no laila ke kiʻekiʻe cholesterol (me ka LDL cholesterol);
- Hoʻonui i ka pale ʻana i ka insulin; a
- Hoʻonui i ka mana glycemic.
Manaʻo nui ʻia ka hopena o ka ʻōpū o ka orlistat i ke ʻano like me ka hoʻoikaika maikaʻi ʻole, e paipai ana i ka poʻe ma kēia lāʻau lapaʻau e pili pono i ka meaʻai haʻahaʻa momona.
(2) Nā CASIDILO CAS: 282526-98-1
ʻO Cetilistat kahi mea hoʻoikaika waha, novel, pancreatic a me gastrointestinal lipase inhibitor. ʻO ka lāʻau hoʻemi kaumaha ʻo Cetilistat he lāʻau lapaʻau i hana ʻia e mālama i ka momona. He hana like ia e like me ka lāʻau i kūkākūkā ʻia ma mua i kapa ʻia ʻo Xenical (orlistat) ma ke kāohi ʻana i ka lipase pancreatic, ka enzyme e wāwahi i nā triglycerides i loko o ko mākou ʻōpū. Me ka loaʻa ʻole o kēia mau enzymes, ʻaʻole e hoʻoheheʻe ʻia nā triglycerides mai kā mākou meaʻai i loko o nā ʻakika momona manuahi e hiki ke hoʻopaʻa ʻia a hoʻoneʻe ʻia mai ke kino me ka ʻole ʻole.
I loko o nā hoʻokolohuaʻokoʻa e pili ana i nā maʻi kūpona me ka maʻi maʻamauʻole 2 a ma nā maʻi kikowaena e noho ana me ka maʻi maʻamauʻo 2. I ka manawa i lawelaweʻia ai ka pahūʻana o ka pauhana kaumaha no nā hebedoma heʻumikumamālua, ua hoʻohaʻahaʻa nuiʻia ke kaumaha o ke kino, ka cholesterol piha, ka liʻiliʻi lipoprotein cholesterol ma muli o ka placebo.
ʻO ka pākēneka o nā mea hōʻeha kūpono e hōʻike ana i ka ho'ēmi ikiʻana o ke kaumaha o ke kino o ka 5 ka nui ma mua o nā lima hana a pau e like me ka placebo. I ka nui o nā maʻi diabetic, ua hoʻohaʻahaʻa nuiʻia nā HbA1c (kiʻekiʻe hemoglobin glycosylated). Ua hōʻikeʻia keʻano palekana o kēia olakino kaumaha ma muli o ka hopena o ka hopena, me ka hopena i ka steatorrhea (keʻano o ka gastrointestinal) me ka hopena iʻoi aku ma mua o ka mea i loko o kolistlist. Ua hōʻoia kokeʻia kēia lāʻau lapaʻau i Iapana e mālama i ka momona me nā pilikia'ē aʻe.
(3) Lorcaserin HCL(Belviq) CAS: 1431697-94-7
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4.Pehea e kūʻai ai i ka pauka paona maikaʻi ma ka pūnaewele?
E like me kaʻikeʻia mai kā mākou kūkākūkā kūkākūkā, nui nā lāʻau'alomolo kaumaha i loaʻa ma laila e laweʻia mai ana mai kahi pūnaeweleʻano nui. ʻO ka hapa nui o kēia mau lāʻau lapaʻau uaʻikeʻia he mea kūpono, a ua'āponoʻia kekahi o lākou e nā mana'ē aʻe e like me FDA a me Iapana, e haʻi aku i kekahi, no ka mālamaʻana i ka momona.
Ma hope o ka hoʻolilo ʻana i nā hola he nui i ka noiʻi ʻana i nā lāʻau hoʻemi kaumaha, ua hiki iā mākou ke ʻike i kekahi mau mea kūʻai maikaʻi loa o 2018 World's Weight Loss Powder Supplements. ʻO kēia mau mea hoʻopihapiha paona kaumaha e komo pū me ka pauka pohō kaumaha orlistat a me ka pauka pohō kaumaha o lorcaserin. ʻAʻole like me nā mea hoʻopihapiha hoʻēmi kaumaha i loaʻa ma kekahi hale kūʻai lāʻau, ʻo kēia mau lāʻau hoʻohaʻahaʻa kaumaha i kuhikuhi ʻia e nā kauka lapaʻau i hala i nā makahiki o ka hoʻāʻo ʻana no ka loaʻa ʻana o kahi hōʻailona mai ka FDA a me kekahi mau ʻāina ʻē aʻe. Manaʻo nui mākou e hoʻāʻo i kēia mau lāʻau lapaʻau no ka mea ua hōʻoia ʻia ʻaʻole maikaʻi wale nō akā palekana no ka hoʻohana.
Hiki iā ʻoe ke nīnau pehea e kūʻai ai i ka pauka pohō kaumaha orlistat pauka a me ka pauka lorcaserin hcl. Nui nā mea hoʻolako pauka pohō kaumaha ma ka pūnaewele a pono e noʻonoʻo i ka mea maikaʻi loa iā ʻoe. Pono ʻoe e noʻonoʻo i ka maikaʻi o nā huahana a inā hiki ke hoʻouna ʻia iā ʻoe ma kahi palekana, inā pono ʻoe e kūʻai i ka pauka pohō kaumaha ma ka nui, pono ʻoe e ʻike inā ʻo kā lākou ʻōnaehana lako a paʻa paha, e noʻonoʻo e pili ana i ka lawe ʻana i ka laʻana kauoha ma mua o ka nui. kauoha, lawe ia e hoao ma ka oihana 3rd- labs a nānā i ka maikaʻi. Eia nō naʻe, ʻaʻole maʻalahi ka loaʻa ʻana o ka mea hoʻolako kiʻekiʻe, pono ʻoe e hoʻonui i ka manawa a me ka ikaika.
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NPP
1. Pehea e kōkua ai ka lorcaserin iāʻoe e lilo i ka kaumaha?
No ka pohō kaumaha, hana ʻo Lorcaserin ma ka hoʻopili ʻana i ke ʻano o ke kino o ka manaʻo piha ma ka hoʻololi ʻana i nā pae serotonin i loko o ka lolo. Ma kēia ala e hiki ai iā Lorcaserin ke hana e mālama i ka addiction opioid.
2. Ua hoʻomaluʻia ka lorcaserin hcl pauka?
ʻOiaiʻaʻole he mea hoʻonāukiuki, hiki i ka lorcaserin ke hana i ka lāʻau lapaʻau a me ka hoʻomāinoino. No kēia kumu, ua hoʻonohonohoʻia e ka Drug Enforcement Administration (DEA) ia ma lalo o ke Kanawai Manaʻo Hoʻoholoʻia ma ka Mokuna IV.
No laila, pehea lā lākou e mālama ai i kahi lāʻau? E wehewehe wau. Hiki paha ke lilo i kahi pohō ka hopena a hiki paha i ka hana e hoʻonāukiuki i ka mea hoʻohana. I mea e lawe ai i kaʻoluʻolu, hiki iāʻoe ke hoʻopiha i nā kauoha no ka palena manawa wale.
ʻO kekahi o nā hopena o ka lorcaserin e komo i loko o ka naʻau, ka manaʻo 'kiʻekiʻe', ka hoʻokaumaha, a me ka euphoria. I kekahi mau kumu, ua hōʻike kekahi mau maʻi i hoʻomaha i ka hōʻailona i kekahi mau hōʻailona haʻalele. ʻO kēia mau mea a pau ka hōʻoia e hiki i ka lāʻau lāʻau ke hoʻonā i ke olaʻana.
3. Ua palekana ka lāʻau paona lorcaserin hcl?
Ua loaʻa i kahi noiʻi nui nā hopena hoʻohiki no ka palekana o kahi lāʻau paona kaumaha i loaʻa i ka US. ʻO ke aʻo ʻana, i paʻi ʻia ma ka New England Journal of Medicine, i ʻōlelo ʻia e nā pākeke e hoʻohana ana i ka lāʻau lorcaserin ua nalowale ka awelika o 4kg (8.8lb) ma luna o 40 mahina. Ua ʻōlelo ʻia ʻo ka lāʻau lapaʻau, e hana ana ma ke kāohi ʻana i ka ʻai, ʻaʻole ia e kau i ka poʻe i ka pilikia nui o nā pilikia naʻau. Akā, hoʻoikaika ka poʻe akamai i ke koʻikoʻi o nā loli ola lōʻihi i ka loaʻa ʻana o ka pohō kaumaha. Ua loaʻa ʻo Lorcaserin ma US no kekahi mau makahiki ma lalo o ka inoa Belviq, akā ʻaʻole i ʻae ʻia no ka hoʻohana ʻana ma ʻEulopa.
4. He kūpono anei ʻo Orlistat no ka pohō kaumaha?
Hana ʻo Orlistat ma ka pale ʻana i ka momona mai ka meaʻai āu e ʻai ai mai ka komo ʻana i loko o kou kino. ʻO kēia momona e puka i waho o ke kino ma o kāu mau fee.
No ka hana ʻana o Orlistat, pono e hoʻohana pū ʻia me nā ʻano hana ʻē aʻe. ʻO kēia mau mea he papahana hoʻoikaika kino maʻamau a me kahi hoʻolālā meaʻai olakino. Ke lawe ʻia iā ia iho, ʻaʻole hiki i Orlistat ke hoʻemi i ke kaumaha, no ka mea, ʻaʻole ia e puhi i ka momona o kēia manawa.
Ua ʻike ʻia kahi haʻawina ʻo ka poʻe i lawe iā Orlistat a mālama i ka meaʻai haʻahaʻa haʻahaʻa i nalowale i ka awelika 1.25 pōhaku (8.1kg) i ka makahiki, ʻo ia ka 6lb (2.8kg) ʻoi aku ka nui o ka poʻe i lawe ʻole iā Orlistat i ka manawa like. Ua ʻike ʻia kahi noiʻi ʻē aʻe he 743 mau maʻi paʻakikī e lawe ana iā Orlistat no ka pohō kaumaha i nalowale ma ka awelika 10.3kg o ke kaumaha ma hope o hoʻokahi makahiki. He ʻokoʻa kēia i ka poʻe maʻi 6.1kg ʻaʻole lawe iā Orlistat nalowale.
Ua ʻike ʻia nā haʻawina ʻē aʻe e hiki i ka poʻe e hahai ana i kēia ʻano lapaʻau ke lilo i 10% o ko lākou kaumaha kino i hoʻokahi makahiki.
5.ʻO wai ka mea e hoʻohana i ka pauka orlistat?
ʻO Orlistat no ka pohō kaumaha ʻoi aku ka maikaʻi e lawe ʻia e ka poʻe e hakakā nei e lilo i ke kaumaha ma o nā ʻano ʻē aʻe. Ma mua o ka hoʻomaka ʻana iā Orlistat, pono ʻoe e hoʻāʻo mua i ka lilo ʻana i ke kaumaha ma o ka ʻai ʻana i ka calorie a me ka hoʻoikaika mau. Pono ʻoe e noʻonoʻo e haʻalele i ka puhi ʻana a me ka hoʻemi ʻana i ka inu ʻana i ka waiʻona ma mua o ka lawe ʻana i ka lāʻau lapaʻau. Ma hope o ka lawe ʻana iā Orlistat no kekahi mau pule, hiki iā ʻoe ke manaʻo e ʻike i ka pohō kaumaha. ʻOkoʻa ka nui maoli ma waena o kēlā me kēia kanaka, ma muli o kā lākou ʻai a me ke ʻano hoʻoikaika kino.
6.Orlistat pauka loiloi: ma mua a ma hope
Zak (4th, Mar. 2021): ʻO kēia ka papahana hoʻoemi kaumaha mua i hiki iaʻu ke paʻa. Paipai nui wau iā Orlistat pauka. Inā ʻaʻole ʻoe makemake i ka "hopena lapaʻau", a laila nānā pono ʻoe i kāu ʻai momona! ʻAʻole hiki iaʻu ke ʻōlelo nui e pili ana i ka pauka Orlistat. Ua ʻike au hiki iaʻu ke loaʻa nā ʻano meaʻai like ʻole - akā ʻo ka nui o ka ʻāpana ke kī!
Jimmy(16, ʻApelila 2020): ʻO nā wiki 3 i kēia manawa maikaʻi loa mai koʻu kūʻai ʻana i ka pauka orlistat ma ka pūnaewele a hoʻāʻo i kekahi. Ke emi nei au i ke kaumaha, ʻo ia kaʻu e makemake ai i loaʻa ʻole iaʻu ka hopena yoyo. E noho ma kāu ʻai haʻahaʻa momona. Ua ʻai au i ka pizza i hoʻokahi lā a hahai aku me ʻelua mau ʻāpana no ka ʻaina kakahiaka a loaʻa iaʻu ka ʻaila ʻalani i ka wā e hele ai ke kinoea a i ka wā o ka ʻōpū. ʻAe e hōʻike iā ʻoe ke ʻai nui ʻoe a i ʻole ka mea hewa. E helu i kāu mau calorie e ʻai i nā mea kanu a me nā hua. E inu wai. Ma hope o ka heluhelu ʻana i nā ʻaoʻao ʻē aʻe, kōkua ia iaʻu e pili pū me Alli no ka mea i ka wā e hiki mai ai, e ʻoki ʻoe i kou poʻo me ka manaʻo UhUh, ʻaʻole, hoʻomākeʻaka ʻoe iaʻu.
Bob(24th, Sep. 2021): Ua lilo au i 6 paona i ka pule hoʻokahi me ka pauka orlistat.. akā ʻai wau i ka meaʻai olakino mon thru fri: ʻai haʻahaʻa momona a haʻahaʻa calories a me ka hopena pule ʻai wau i kekahi mea maʻalahi. Eia kekahi, hele au i 45 mau minuke i kēlā me kēia lā a pāʻani i ka tennis 3 mau hola ma ka noho.
E like me ka hōʻike ʻana o nā loiloi ma luna nei, ʻoi aku ka maikaʻi o ka ʻike o kā mākou mea kūʻai aku iā Orlistat ma ke ʻano he mālama kaumaha. Eia kekahi o nā kumu nui i hōʻike ʻia e kā mākou mea kūʻai aku iā Orlistat:
♦ He kūpono ia i ke kōkua ʻana i nā maʻi e hoʻemi i ke kaumaha
♦ He mea maikaʻi ia no ka hoʻomaka ʻana i kahi hoʻolālā hoʻemi kaumaha
♦ He mea maikaʻi ia no ka hoʻohaʻahaʻa paona i kēlā me kēia pule
♦ He mea pono no ka hoemi ana i ka cholesterol
Ma ke ʻano holoʻokoʻa, kuhikuhi kā mākou mea kūʻai aku iā Orlistat ma ke ʻano he ala hilinaʻi a maikaʻi hoʻi e lilo ai ke kaumaha.
7. He aha nā hopena o ka orlistat?
Nā hopena maʻamau o Orlistat
ʻO nā hopena ʻaoʻao maʻamau o Orlistat e pili pinepine i hoʻokahi ma 10 poʻe. Aia kēia mau mea i lalo, akā ʻo ka hopena maʻamau ka maʻi poʻo:
▪ ʻAila a momona paha a i ʻole ka ʻaila mai kou anus - e nānā i nā wahi ʻaila ma kou lole komo.
▪ Kokoke a i ʻole ka hoʻonui ʻana i ka ʻōpū
▪ Hoʻonui ʻia ka ʻōpū, i kekahi manawa me ka hoʻokuʻu ʻana
▪ Poʻomanaʻo poʻo
▪ ʻO nā maʻi ʻeha o ka ʻōpū o luna (RTI), e like me ke anu
▪ ʻEha o ka ʻōpū a ʻeha paha
He manawa pōkole kēia mau hopena a pono e hala me ka manawa. Eia naʻe, inā ʻike ʻoe iā lākou no ka manawa lōʻihi, a i ʻole e ʻoi aku ka ʻino, e kamaʻilio koke me kāu kauka.
ʻO nā hopena ʻaoʻao maʻamau o Orlistat
ʻO nā hopena ʻaoʻao o Orlistat ma lalo nei he mea maʻamau ia ma mua o nā mea i helu ʻia ma luna a me:
▪ ʻO nā faeces palupalu
▪ Ka hoʻomau ʻole ʻana o ka fecal
▪ Nā maʻi ʻāʻī a i ʻole nā niho
▪ ʻO ka ʻūhā — ʻoi aku ka maʻamau o kēia i ka poʻe me ka maʻi maʻi type 2
▪ Nā wā kūpono ʻole
▪ Luhi
▪ ʻO nā maʻi hanu haʻahaʻa
▪ Ka ʻeha a i ʻole ka hōʻoluʻolu
Inā ʻike ʻoe i kekahi o kēia mau hopena ʻaoʻao no kahi manawa lōʻihi a i ʻole e hoʻomaka ana kāu mau hōʻailona e ʻino, e kamaʻilio me kāu kauka i ka wā hiki.
8. Pehea e hiki ai iaʻu ke hoʻemi i nā hopena o Orlistat?
ʻO ka hapa nui o nā hopena ʻaoʻao o Orlistat he manawa pōkole a hele me ka manawa. Inā ʻaʻole i pau nā hopena ʻaoʻao, e kamaʻilio me kāu kauka i ka hikiwawe. Hiki ke hōʻemi i nā hopena ʻaoʻao o Orlistat ma ke ana ʻana i ka nui o ka momona āu e ʻai ai i kēlā me kēia pāʻina.
Hana ʻo Orlistat ma ke kāpae ʻana i nā momona i kāu meaʻai mai ka komo ʻana i loko o ka ʻōpū. Hoʻokuʻu aku ia i nā momona ʻaʻole i lawe ʻia ma ka ʻōpū. Eia naʻe, hiki iā Orlistat ke hoʻopau wale i ka momona nui i kēlā me kēia ʻai. No laila, inā ʻoe e ʻai i ka meaʻai me ka ʻoi aku o ka 1-15 grams o ka momona, hiki iā ʻoe ke ʻike pinepine i nā hopena ʻaoʻao o Orlistat. No ka hōʻemi ʻana i nā hopena ʻaoʻao o Orlistat, ʻaʻole ʻoi aku ma mua o 1-15 grams o ka momona i kēlā me kēia pāʻina inā ʻoe e lawe iā Orlistat 120 mg capsules.
Hiki iā ʻoe ke hōʻemi i nā hopena ʻaoʻao o Orlistat ma ka hoʻopili ʻana i ke ʻano kūpono o Orlistat. ʻO ka lawe ʻana i nā mea i ʻōlelo ʻia ma Orlistat ma hope o ka ʻai ʻana e hoʻonui i kona hopena ʻaoʻao, no laila e hoʻopili i ka dosage i ʻōlelo ʻia.
9.How e hoʻolālā i ka palahalaha Palekana e mālama ai i ka nui?
ʻO ka uluʻana o ka momona ua hoʻonāukiuki i ka huliʻana i nā lāʻau lapaʻau e mālama i kēiaʻano. Ua nānā 'ia nā' ano lapaʻauʻokoʻa, e like me:
▪ Serotonin a me ka noradrenaline reuptake inhibitors (anorectic agents)
▪ Nā mea pale lipase
▪ b 3-adrenoreceptor agonists
▪ ʻO nā agonists leptin
▪ ʻO nā agonists melanocortin-3
▪ Endocannabinoid receptor antagonists
ʻO ka pauka Cetilistat he mea lipase inhibitor, me keʻano like o ka hana i ka lāʻau anti-obesity o Roche orlistat pauka i loaʻa i ka'āpono hoʻoponopono i ka 1997. Ke hana nei kēia mau lāʻau lapaʻau i ka'ōpū o ka'ōpū e pale i nā lipases, nā enzymes i komo i ka hakiʻana o nā momona meaʻai. Ma ke kāohi ʻana i ka haʻihaʻi a me ka komo ʻana o nā momona mai ka ʻōpū, hoʻemi ka lipase inhibitors i ka momona momona a me nā calorie, no laila e kōkua ai i ka lilo ʻana o ka momona.
10.Orlistat Powder Vs Cetilistat pauka
mau | Pauka Orlistat | Paleheʻe kēiailistat |
Ka helu CAS | 96829-58-2 | 282526-98-1 |
Ka hana hana | ʻAʻole hana ʻo Orlistat ma ke kāohi ʻana i ka ʻai; e hoemi ana i ka nui o na momona a kou kino e komo ai mai ka ai au e ai ai. | ʻO Cetilistat kahi mea hoʻopaneʻe lipase gastrointestinal e hoʻopaʻa ana i ka momona momona a me ka absorption, e alakaʻi ana i ka hoʻemi ʻana i ka ikehu, a no laila ke pohō kaumaha. |
Hoʻoponopono | 120 mg i ka waha ʻekolu manawa i ka lā me kēlā me kēia ʻai nui i loko o ka momona. | 120 mg ʻekolu manawa i ka lā ma hope koke o kēlā me kēia ʻai. |
Nā hopenaʻaoʻao | ▪ Ke kinoea holo kino, i kekahi manawa me ka ʻaila ▪ ʻO nā peʻa maloʻo, nā pehu momona, a i ʻole ka maʻi maʻi ▪ ʻO ka ʻōpū pinepine a i ʻole ka neʻe ʻana o ka ʻōpū paʻakikī ke hoʻomalu ▪ Kaohi paʻa ▪ ʻeha ʻōpū ▪ Pupuu | ▪ Aila ▪ ʻO nā ʻūhā maloʻo ▪ Ka hoʻomau ʻole ʻana o ka fecal ▪ Ka ʻūhā ▪ ʻEha ʻōpū ▪ Nā ʻūhā palupalu ▪ Waha Maloo
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Reviews | ☆☆☆☆ | ☆☆☆ |
Reference
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