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Hexarelin

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Nā inoa'ē aʻe:phenylalanyl-L-lysinamide

ʻO AASraw ka mea hanaʻoihana o peptide Hexarelin nona ka hale kūʻokoʻa kūʻokoʻa a me ka hale hana nui e like me ke kākoʻo, e hanaʻia nā hana a pau ma lalo o ke kānāwai CGMP a me ka pūnaewele mana o ka maikaʻi. nā hue.

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Product Description

He aha ka Hexarelin?

Ma muli o ka hiki iā Hexarelin ke hoʻonui i ka huna ʻana o ka Hormone Growth maoli, ʻo ka hapa nui o kāna mau hopena e like me ka GH synthetic, ʻoiai i kahi liʻiliʻi liʻiliʻi. ʻO ka nui o nā ʻiʻo ʻiʻo i loaʻa i kēia manawa, ka pale neural, ka hui hou ʻana, ka pale a me ka ho'ōla. Eia kekahi, ʻo nā mea loaʻa GH i loko o ka ʻiʻo adipose (momona) hiki ke hoʻemi i ka momona me ka hoʻohana ʻana iā Hexarelin. -E like me Growth Factor (IGF-1) e piʻi i loko o ke akepaʻa. ʻO IGF-1 ke kumu nui o ka ulu ʻana o ka ʻiʻo ma ka pane ʻana i ka hoʻoulu ʻana o GH.

ʻAʻohe mea e hoʻonui ai i ka makemake me ka hoʻohana ʻana iā Hexarelin (e kūʻē i ka piʻi ʻana o ka makemake nui o GHRP-6) ma muli o kona hiki ʻole ke hoʻonui nui i nā pae Ghrelin i kuleana no ka pōloli hou a me ka wikiwiki o ka hoʻokuʻu ʻana i ka ʻōpū.

Ma nā haʻawina kahi i hoʻokomo ʻia ai ʻo Hexarelin subcutaneously, Growth Hormone, i ana ʻia ma ka plasma concentrations, piʻi nui ʻia a i loko o kanakolu mau minuke o ka injection. Ua emi hou nā pae GH i ka maʻamau ma kahi o ʻehā mau hola ma hope o ka injection. Ua ʻike ʻia ka piʻi ʻana o ka GH a hiki i 2mg/ kg, ua ʻike ʻia ʻaʻole pono ka hoʻonui hou ʻana o ka maʻi i ka hana ʻana i ka pane GH.

Ua hōʻike ʻia ka noiʻi ua emi ka hopena o Hexarelin i ka hoʻoulu ʻana i ka GH ma waena o nā pule 4 a hiki i 16. ʻO ka hoʻokaʻawale ʻana i nā pōʻai ma nā wiki he 4 o nā manawa, e pale ana i ka puka manaʻo maikaʻi ʻole a me ka pōʻai hou o Hexarelin i hoʻopuka i ka pae o nā hopena e like me ka pōʻai mua.

Hexarelin (Hexarelin Acetate) he hexapeptide synthetic i loko o ka ʻohana ulu ulu e hoʻoulu ai i ka hoʻokuʻu ʻana o ka hormone ulu (GH) a ʻaʻole keakea i ka hiki o ke kino ke hana i kāna iho GH. ʻO GHRP-6 akā me ka ʻole o ka hoʻonui ʻana i ka makemake ma muli o kona hiki ʻole ke hoʻonui nui i nā pae Ghrelin nona ke kuleana no ka hoʻonui ʻana i ka ʻai a me ka wikiwiki o ka hoʻokuʻu ʻana o ka ʻōpū. ʻO ke kino kanaka.Hexarelin i loko o nā haʻawina i kekahi manawa ua hōʻike ʻo ia e hōʻemi i ka momona visceral.Hexarelin (Hexarelin Acetate) e like me nā mea ʻē aʻe Growth Hormone Releasing Peptides ʻoi aku ka maikaʻi synergistically ke lawelawe ʻia me GHRH e like me Sermorelin a i ʻole Modified GRF 1-29.

Pehea ka hana o Hexarelin?

ʻO ka Hexarelin mai AASraw ʻaʻole ia e like me nā GHRP ʻē aʻe i loaʻa i kēia lā. Manaʻo ka poʻe he hexarelin ma ke ʻano he underdog. he peptide i hoʻohaʻahaʻa ʻia. I kēia lā, eia naʻe, e haʻi mākou iā ʻoe i ke kumu e pono ʻole ai e kāpae ʻia kēia peptide kikoʻī.

Pono ʻoe e ʻike ʻaʻole ʻo ka hexarelin kāu GHRP maʻamau. ʻO kona ʻano he hexapeptide he ala maikaʻi loa ia e hāpai i ka hoʻonui ʻia ʻana o nā hormones ulu. ma ka ʻāpana hypothalamic a me ka pituitary gland. ʻO ka mea nui, ʻo ia ka peptide hoʻokahi e hiki ke hana i ka nui o nā hormones ulu.

E like me ka nui o nā peptides, hiki i ka hexarelin ke hoʻonui i ka hoʻokuʻu ʻana o nā hormones ulu maoli. ʻO ka mea nui, ʻaʻole ia e hoʻemi i ka hiki maoli o ke kino e hoʻokuʻu i nā hormones ulu. hoʻomaikaʻi i ka elasticity o ka ʻili a hoʻonui i ka mitosis, meiosis a me ka iwi mineral density.

Eia naʻe, ua hōʻike ʻia nā haʻawina i ka manawa i hoʻopaʻa ʻia ai ka hexarelin ma ke ala subcutaneous, hoʻāla ia i ka hana o ka pituitary gland ma o ka pulse. Like me GHRP-6, kōkua ia i ka hoʻomaikaʻi ʻana i ke kahe o nā hormones ulu i loko o ke kino. ʻO GHRP-6, he hana ʻokoʻa ia ma kekahi mau ʻano. No ka mea hoʻokahi, ʻaʻole ia e hoʻopilikia i ka pōloli. nā kumu nui o ka hanaʻoleʻana i nā hormones ulu.

Me kona hiki ke hoʻokiʻekiʻe i ka IGF-1 a me ke kiʻekiʻe o ka hormone ulu, hiki iā ia ke hana ma ke ʻano he mea hana PCT maikaʻi loa no nā poʻe e holo kaʻa me ka synthetic IGF-1 a i ʻole nā ​​​​hormone ulu ʻē aʻe. hoʻonui i nā pae o ka prolactin a me ka cortisol. Loaʻa iā ia ka pilina ikaika loa e hoʻonui i ka cortisol a me ka prolactin i hoʻohālikelike ʻia me nā GHRP i loaʻa.

ʻO nā pono o Hexarelin

①Ka Ulu ʻana o ka ʻiʻo Lean

ʻAʻole ʻoe wale nō inā hauʻoli ʻoe i kou paona a i ʻole ke ʻano o ke kino. Akā naʻe, ʻaʻole maʻalahi ka loaʻa ʻana o kahi kumulāʻau palekana a hilinaʻi no ka loaʻa ʻana o ka ʻiʻo lean. ke ano e hoao ana e lapaau.

ʻO ka mea pōmaikaʻi, ua hoʻohiki ka noiʻi mua ma Hexarelin a he nui ka poʻe e kū nei ma hope o ka peptide i ke kaiāulu hāpai kaumaha. Ua ʻike ʻia ʻo Hexarelin e hoʻoulu i ka ulu ʻana o ka hormone ulu maoli e kōkua i ka ulu ʻana o ka ʻiʻo lean. -like Growth Factor 1 (IGF-1) He hana like ia me ka ghrelin i ka hoʻoulu ʻana i ka hormone ulu ulu secretagogue receptor aʻo ka hoʻopau ʻana i nā inhibitors e like me somatostatin. ʻO ka poʻe e hoʻohana ana iā Hexarelin i ka hoʻoikaika kino a me ke bodybuilding e hoʻomaopopo i nā hopena kupaianaha e pili ana i ka loaʻa ʻana o ka ʻiʻo a me ka ikaika.

②Ke puhi momona a me ke kaumaha

Hiki ke kūkulu i ka ʻiʻo wīwī ma ka wehe mua ʻana i ka momona i makemake ʻole ʻia.

ʻO ka mea pōmaikaʻi, hiki iā Hexarelin ke hoʻoikaika i ka pohō kaumaha ma ka huli ʻana i nā kaʻina kūlohelohe koʻikoʻi i loko o ke kino. ʻO ka hopena o ka momona momona hiki ke kōkua iā ʻoe i ka hoʻokō ʻana i kāu mau pahuhopu kaumaha ma mua o ka wā. ʻO ka hui pū ʻana o ka momona momona a me ka loaʻa ʻana o nā ʻiʻo lean mai Hexarelin hiki ke alakaʻi i kahi hoʻoponopono kino piha.

③ Hoʻomaikaʻi i ka ikaika a me ka maʻalahi

ʻOiai e loaʻa ana i kahi hoʻololi kino holoʻokoʻa, loaʻa iā ʻoe nā pōmaikaʻi o ka hoʻomaikaʻi ʻana i ka ikaika a me ka maʻalahi.

ʻIke ʻia ʻo Hexarelin e hoʻomaikaʻi nui i ka tendon a me ka ikaika ligament. Eia kekahi, pili ka peptide i ka hoʻonui ʻia a me ke olakino hui holoʻokoʻa.

No laila, hiki iā ʻoe ke hoʻokō liʻiliʻi inā paʻa ʻoe ma ka ʻaoʻao ma muli o kahi hōʻeha mau.

④ʻoi aku ka ikaika o ka hoʻihoʻi hou ʻana a me ka hana haʻuki

Loaʻa nā pōmaikaʻi hou i ka lilo ʻana o ke kaumaha, ka loaʻa ʻana o ka ʻiʻo lean, a me ka hoʻomaikaʻi ʻana i ka ikaika holoʻokoʻa.

No ka hoʻomaka ʻana, e hoʻōla wikiwiki ʻoe e hāʻawi iā ʻoe i ka manawa e hoʻi ai i ka hale haʻuki a hoʻi i ka hana. He mea nui ka hoʻihoʻi ʻana i ka pohō kaumaha a me ka loaʻa ʻana o ka ʻiʻo, no laila he mea nui ka loaʻa ʻana o nā mea hoʻohui e kōkua i kēlā kaʻina hana.

ʻIke ʻia ʻo Hexarelin e hāpai i ka hoʻōla wikiwiki ʻana mai nā ʻeha a me ka hoʻomaʻamaʻa.

Eia kekahi, e ʻike ʻoe i ka holomua holoʻokoʻa o ka hana haʻuki ma muli o ka hopena.

⑤ Hoʻomaikaʻi i ka maikaʻi o ka hiamoe a me ka maikaʻi holoʻokoʻa

ʻO kekahi pōmaikaʻi ʻē aʻe iā Hexarelin he mau hōʻike e pili ana i ka hoʻomaikaʻi ʻana o ka peptide i ka maikaʻi o ka hiamoe holoʻokoʻa.

A, no ka mea, he mea nui ka hiamoe i ke olakino holoʻokoʻa, hāʻawi ka peptide i ka manaʻo maikaʻi aʻe.

ʻAʻole wale ʻoe e hiamoe maikaʻi akā ʻoi aku ka maikaʻi o ka mahalo i nā hopena maikaʻi o Hexarelin.

Nā hopena ʻaoʻao o Hexarelin

Mahalo, ʻaʻole liʻiliʻi nā hopena ʻaoʻao o Hexarelin.

ʻO nā hopena ʻaoʻao maʻamau ka manaʻo o ka luhi a i ʻole ka lethargy. Ma muli o ka hiki o ka hormone ulu e hoʻonui i ka makemake no ka hiamoe. Akā naʻe, ʻo ka mālama ʻana i ka haʻahaʻa haʻahaʻa hiki ke hoʻopau i kēia pilikia. paʻa wai.

ʻO kekahi hopena ʻaoʻao i hōʻike ʻia ʻo ke kani ʻana a i ʻole ka helu ʻana i nā lima a i ʻole nā ​​wāwae.

ʻO ka poʻe i ʻike i nā hōʻailona e hoʻohaʻahaʻa i ka dosage a i ʻole e noʻonoʻo e wehe i ka supplementation a pau.

ʻOi aku ka maikaʻi e kamaʻilio me ke kauka ma mua o ka hoʻohana ʻana inā ua lawe mua ʻoe i nā lāʻau lapaʻau ʻē aʻe.

Hexarelin me nā peptides ʻē aʻe

Hexarelin vs Ipamorelin

ʻOiai ke ʻano o ka hana a me nā pono mua no nā peptides ʻelua, ʻokoʻa ka ʻokoʻa i nā pono lua.

Hexarelin vs GHRP-6

Hoʻohana like kēia mau peptides ʻelua. Akā naʻe, ʻaʻole maʻalahi ka GHRP-6 (9) i ka hoʻoulu ʻana i nā ala neuroendocrine ʻē aʻe e like me hexarelin. .No laila, lanakila ʻo hexarelin i ka heihei kūʻē iā GHRP-6 no ka maopopo!

Ma hea e kūʻai ai i ka Hexarelin?

He hopena koʻikoʻi ka Hexarelin peptide therapy i ke olakino holoʻokoʻa. Kōkua ia i ka loaʻa ʻana o ka ʻiʻo, ka metabolizing momona, ka hoʻonui ʻana i ka ikehu, a me nā mea ʻē aʻe. Eia ma AASraw, ua hoʻolaʻa mākou i ka hāʻawi ʻana i nā peptide he nui e pili ana i ka pohō kaumaha, nā mālama ola kino, a me nā mea ʻē aʻe. hormone.Inā makemakeʻoe i ka Hexarelin nui a iʻole nā ​​peptides'ē aʻe, e hoʻopiha i ka hōpili ma lalo nei e hoʻonohonoho i kāu kūkākūkā a kamaʻilio me kā mākou limahana kūikawā.ʻAʻole hiki iā mākou ke kali e lohe mai iāʻoe!

Hexarelin Hōʻike Hōʻike-HNMR

He aha ka HNMR a He aha ka HNMR spectrum e haʻi aku iā ʻoe? ʻO H Nuclear Magnetic Resonance (NMR) spectroscopy kahi ʻenehana kemika analytical i hoʻohana ʻia i ka hoʻokele maikaʻi a me ka noiʻi no ka hoʻoholo ʻana i ka ʻike a me ka maʻemaʻe o kahi laʻana a me kona ʻano molekala. No ka laʻana, hiki i ka NMR ke hoʻokaʻawale i nā hui pū ʻia i ʻike ʻia. No nā pūhui i ʻike ʻole ʻia, hiki ke hoʻohana ʻia ka NMR e hoʻohālikelike i nā hale waihona puke spectral a i ʻole e kuhi pololei i ke ʻano kumu. Ke ʻike ʻia ke ʻano kumu, hiki ke hoʻohana ʻia ka NMR no ka hoʻoholo ʻana i ka conformation molecular i ka hopena a me ke aʻo ʻana i nā waiwai kino ma ka pae molekala e like me ka hoʻololi conformational, nā hoʻololi ʻana, ka solubility, a me ka diffusion.

Pehea e kūʻai ai iā Hexarelin mai AASraw?

❶E hoʻokaʻaʻike mai iā mākou ma kā mākou ʻōnaehana nīnau leka uila, a i ʻole e waiho i kāu helu whatsapp iā mākou, e hoʻopili aku kā mākou mea kūʻai aku (CSR) me ʻoe i 12 mau hola.

❷E hāʻawi mai iā mākou i kāu helu a me kāu helu wahi i nīnau ʻia.

❸Na kā mākou CSR e hāʻawi iā ʻoe i ka ʻōlelo, ka manawa uku, ka helu ʻimi, nā ala hoʻouna a me ka lā i manaʻo ʻia (ETA).

❹E uku ʻia a hoʻouna ʻia nā waiwai i loko o 12 mau hola.

❺ Loaʻa nā waiwai a hāʻawi i nā manaʻo.

Mea kākau o kēia ʻatikala:
Kauka Monique Ua puka 'o Hong mai ke Kula Nui o UK Imperial College London Faculty of Medicine

Mea kākau moʻolelo puke moʻolelo ʻepekema:
1. David Dahlgren
mahele o Pharmaceutical Biosciences, Translational Drug Discovery and Development, Uppsala University, Uppsala 752 36, Suedena
2. H. McDonald
Kula o Biomedical Science, University of Queensland, Brisbane, Australia
3. Giuseppe Biagini
Laboratory of Experimental Endocrinology, Department of Internal Medicine, The Sahlgrenska Academy ma ke Kulanui o Gothenburg, Gothenburg, Suedena
4. Anna Barlind
Keʻena o ka Psychiatry, University of Medicine and Dentistry of New Jersey, Robert Wood Johnson Medical School, Piscataway, NJ, USA
ʻAʻole ʻae kēia kauka/ ʻepekema i ke kūʻai, kūʻai ʻana, a hoʻohana paha i kēia huahana no kekahi kumu. ʻAʻohe pili a pili ʻole ʻo Aasraw, i hōʻike ʻia a i ʻole, me kēia kauka. ʻO ke kumu o ka haʻi ʻana i kēia kauka, ʻo ia ka hoʻomaikaʻi, hoʻomaikaʻi a hoʻomaikaʻi i ka hana noiʻi a me ka hoʻomohala piha i hana ʻia e nā ʻepekema e hana nei i kēia mea.

E hoʻomaopopo '

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[2] Ezio Ghigo (1999). Growth Hormone Secretagogues: Nā ʻike kumu a me nā hopena lapaʻau. Elsevier. aoao 178–. ISBN 978-0-444-82933-7.

[3] Rahim A, O'Neill PA, Shalet SM (1998). "Ke kūlana hormone ulu i ka wā lōʻihi hexarelin therapy". ʻO ka Journal of Clinical Endocrinology & Metabolism. 83 (5): 1644–9. doi:10.1210/jcem.83.5.4812. PMID 9589671.

[4] Ghigo E, Arvat E, Gianotti L, Imbimbo BP, Lenaerts V, Deghenghi R, et al. (1994). "Ka hana hoʻokuʻu ʻana i ka hormone ulu o hexarelin, he hexapeptide synthetic hou, ma hope o ka intravenous, subcutaneous, intranasal, a me ka hoʻokele waha i ke kanaka". ʻO ka Journal of Clinical Endocrinology & Metabolism. 78 (3): 693–8. doi:10.1210/jcem.78.3.8126144. PMID 8126144.

[5] Imbimbo, BP; Mant, T.; Edwards, M.; Amin, D.; Dalton, N.; Boutignon, F.; Lenaerts, V.; Wďż˝thrich, P.; Deghenghi, R. (1994). "Ka hana hoʻokuʻu ʻana i ka hormone ulu o ka hexarelin i nā kānaka". European Journal of Clinical Pharmacology. 46 (5): 421–5. doi:10.1007/bf00191904. PMID 7957536. S2CID 19573322.

[6] CR Ganellin; ʻO David J. Triggle (21 Nowemapa 1996). ʻO ka puke wehewehe ʻōlelo o nā Agena Pharmacological. CRC Press. aoao 617–. ISBN 978-0-412-46630-4.


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