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Hexarelin

Rating: Māhele:

Nā inoa'ē aʻe:phenylalanyl-L-lysinamide

ʻO AASraw ka mea hanaʻoihana o ka peptide Hexarelin nona ka lab kūʻokoʻa a me ka hale hana nui e like me ke kākoʻo, e hoʻokō ʻia nā hana āpau ma lalo o ka hoʻoponopono CGMP a me ka ʻōnaehana mālama maikaʻi trackable. Hiki iā AASraw ke ʻae i ka lawelawe maʻamau e like me nā noi kikoʻī ma peptide pauda maka a pau paha nā hue peptide.

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Kauoha Nui

Product Description

He aha ka Hexarelin?

Ma muli o ka hiki iā Hexarelin ke hoʻonui i ka huna ʻana o ka Hormone Growth maoli, ʻo ka hapa nui o kāna mau hopena e like me ka GH synthetic, ʻoiai he liʻiliʻi iki. ʻO nā hopena o kona hoʻohana ʻana, ʻo ia ka piʻi ʻana o ka ikaika, ka ulu ʻana o nā ʻiʻo ʻiʻo hou, ka hoʻonui ʻana i ka nui o nā ʻiʻo i loaʻa i kēia manawa, ka pale neural, ka hou ʻana o ka hui, ka pale, a me ka ho'ōla. Eia kekahi, ʻae nā mea loaʻa GH i ka kiko adipose (momona) no ka hoʻemi ʻana i ka momona me ka hoʻohana ʻana iā Hexarelin. ʻO ka piʻi ʻana o ka GH kaʻapuni ma o ka hoʻohana ʻana iā Hexarelin ke kumu e piʻi ai nā pae o ka Insulin-Like Growth Factor (IGF-1) i loko o ke ake. ʻO IGF-1 ke kumu nui o ke ulu i ka pane ʻana i ka hoʻoulu ʻana o GH.[3][5]

ʻAʻohe mea e hoʻonui ai i ka makemake me ka hoʻohana ʻana iā Hexarelin (e kūʻē i ka piʻi ʻana o ka makemake nui o GHRP-6) ma muli o kona hiki ʻole ke hoʻonui nui i nā pae Ghrelin i kuleana no ka pōloli hou a me ka wikiwiki o ka hoʻokuʻu ʻana i ka ʻōpū.

I nā haʻawina kahi i hoʻokomo ʻia ai ʻo Hexarelin subcutaneously, Growth Nā Hormone, ana ma o ka plasma concentrations, hoonui nui i loko o kanakolu minuke o ka injection.GH pae ho'ēmi hoʻi i ka maʻamau ma kahi o eha hola ma hope-injection. Ua ʻike ʻia ka piʻi ʻana o ka GH a hiki i ka 2mg/kg, ʻike ʻia kekahi hoʻonui hou ʻana i ka hopena i ʻike ʻole ʻia i ka hopena o ka pane GH.

Ua hōʻike ʻia ka noiʻi ʻana ua emi ka hopena o Hexarelin i ka hoʻoulu ʻana i ka GH ma waena o nā pule 4 a hiki i 16. ʻO ka hoʻokaʻawale ʻana i nā pōʻai ma nā wiki he 4, e pale ana i ka loop manaʻo maikaʻi ʻole, a ʻo ka pōʻai hou o Hexarelin i hoʻopuka i ka pae o nā hopena e like me ka pōʻai mua.

Hexarelin (Hexarelin Acetate) he hexapeptide synthetic i loko o ka ʻohana kumu ulu e hoʻoulu ai i ka hoʻokuʻu ʻana o Ka hormone ulu (GH) a ʻaʻole keakea i ka hiki o ke kino ke hana i kāna GH ponoʻī. Ma ke ano o ka hana, ua like ke ano o Hexarelin (Hexarelin Acetate). GHRP-6 akā me ka piʻi ʻole o ka ʻai ma muli o kona hiki ʻole ke hoʻonui nui i nā pae Ghrelin ke kuleana no ka hoʻonui ʻana i ka ʻai a me ka wikiwiki ʻana o ka ʻōpū. ʻO Hexarelin kahi mea huna hormone ulu synthetic i hana ʻia mai ʻeono amino acids. Loaʻa i ka mana mea hoʻokuʻu hormone ulu i loko o ke kanaka kino. Ua hōʻike ʻo Hexarelin i nā haʻawina i kekahi manawa e hōʻemi ana i ka momona visceral. Hexarelin (Hexarelin Acetate) e like me nā mea ʻē aʻe Ka Hoʻonui Hormone ʻO ka hoʻokuʻu ʻana i nā Peptides ʻoi aku ka maikaʻi me ka synergistically ke lawelawe ʻia me GHRH e like me Sermorelin a i ʻole Modified GRF 1-29.

Pehea ka hana o Hexarelin?

Hexarelin mai KANAKA ʻAʻole like ia me nā GHRP ʻē aʻe i loaʻa i kēia lā. Manaʻo ka poʻe he hexarelin ma ke ʻano he underdog. ʻO ia kekahi o nā mea i loaʻa ʻole i ka nānā ʻana no ka mea ua manaʻo ʻia ʻaʻole nele kekahi mau ʻano koʻikoʻi e pono ai nā peptides maikaʻi loa. Ua lawa ka ʻōlelo ʻana he peptide ka hexarelin i hoʻohaʻahaʻa ʻia. I kēia lā, akā, e haʻi mākou iā ʻoe i ke kumu o kēia kikoʻī ʻakika'amino ʻaʻole pono e hoʻokuʻu ʻia.

Pono ʻoe e ʻike ʻaʻole ʻo hexarelin kāu GHRP maʻamau. ʻO kona ʻano he hexapeptide e hana ia i kahi ala maikaʻi loa e hāpai i ka hoʻonui ʻana i ka hoʻokuʻu ʻana o nā hormones ulu. ʻOiai ʻaʻole i hoʻomaopopo piha ʻia kāna ʻano hana e ka poʻe akamai, ua ʻike ʻia e hana ia ma ka ʻāpana hypothalamic a me ka pituitary gland. ʻO ka mea nui, ʻo ia ka peptide hoʻokahi e hiki ke hana i ka nui o nā hormones ulu.

E like me ka hapa nui o nā peptides, hiki i ka hexarelin ke hoʻonui i ka hoʻokuʻu ʻana o nā hormone ulu maoli. ʻO ka mea nui, ʻaʻole ia e hoʻemi i ka hiki maoli o ke kino e hoʻokuʻu i nā hormone ulu. Ua hōʻike pū kekahi mau haʻawina e hoʻonui i ka momona momona, hoʻoikaika i nā ʻiʻo pili, hoʻomaikaʻi i ka elasticity o ka ʻili, a hoʻonui i ka mitosis, meiosis, a me ka iwi mineral density.

Ua hōʻike naʻe nā haʻawina i ka manawa i hoʻopaʻa ʻia ai ka hexarelin ma ke ala subcutaneous, hoʻāla ia i ka hana o ka pituitary gland ma o ka pulse. E like me GHRP-6, kōkua ia i ka hoʻomaikaʻi ʻana i ke kahe o nā hormones ulu i loko o ke kino. ʻOiai ka loaʻa ʻana o nā mea like me GHRP-6, ʻokoʻa ka hana ma kekahi mau ʻano. ʻO ka mea hoʻokahi, ʻaʻole ia e hoʻopilikia i ka pōloli. Heʻoiaʻiʻo hiki i ka hexarelin ke hoʻonui i ka pae o ka hormone ulu i loko o ke kino, akā hiki ke hoʻemi i ka somatostatin-kekahi o nā kumu nui o ka hana ʻole o nā hormones ulu. ʻO kēia keʻano e hoʻonuiʻia nā kiʻekiʻe o nā hormones ulu.[2][5]

Me kona hiki ke hoʻokiʻekiʻe i ka IGF-1 a me nā pae hormone ulu, hiki ke hana ma ke ʻano he mea maikaʻi loa ʻO ka mea hana PCT no ka poʻe e holo kaʻa ʻO ka IGF-1 synthetic a i ʻole nā ​​​​hormone ulu ʻē aʻe. ʻOi aku ka maikaʻi o nā mea hoʻohana ʻaʻole e hoʻohaʻahaʻa i kona ikaika, ʻoi aku ka nui o ka piʻi ʻana o ka prolactin a me cortisol. Loaʻa iā ia ka pilina ikaika loa e hoʻonui i ka cortisol a me ka prolactin i hoʻohālikelike ʻia me nā GHRP i loaʻa.

ʻO nā pono o Hexarelin

①Ka Ulu ʻana o ka ʻiʻo Lean

ʻAʻole ʻoe hoʻokahi inā manaʻo ʻoe ʻaʻole hauʻoli i kou kaumaha a i ʻole ke ʻano o ke kino. Eia naʻe, ʻaʻole maʻalahi ka loaʻa ʻana o kahi kumulāʻau palekana a hilinaʻi no ka loaʻa ʻana o ka ʻiʻo lean. Nui nā lāʻau lapaʻau ma ka mākeke a ʻoi aku ka ʻino o kekahi o lākou aoao waiwai ma mua o ke kūlana e ho'āʻo nei e mālama.

ʻO ka mea pōmaikaʻi, ua hoʻohiki ka noiʻi mua ma Hexarelin a he nui ka poʻe e kū nei ma hope o ka peptide i ke kaiāulu kaumaha.[4] ʻIke ʻia ʻo Hexarelin e hoʻoulu i ka ulu ʻana o ka hormone ulu maoli e kōkua i ka ulu ʻana o ka ʻiʻo lean.[4] Hoʻohana ka peptide ma ke ʻano he agonist koho nui o ka GHSR a me ka Insulin-like Growth Factor 1 (IGF-1).[6] Hoʻohālikelike ia me ka ghrelin i ka hoʻoulu ʻana i ka ulu ʻana o ka hormone secretagogue receptor aʻo ke kāohi ʻana i nā inhibitors e like me somatostatin. ʻO ka poʻe e hoʻohana ana iā Hexarelin i ka hoʻoikaika kino a me ke bodybuilding e ʻike i nā hopena maikaʻi loa e pili ana i ka loaʻa ʻana o ka ʻiʻo a me ka ikaika.

②Ke puhi momona a me ke kaumaha

Hiki ke kūkulu ʻia ka ʻiʻo lean ma ka wehe mua ʻana i ka momona i makemake ʻole ʻia. He pilikia ka nui o mākou e hakakā nei i ka wā e hoʻāʻo nei e mālama i ka ʻai olakino a me nā hana hoʻoikaika kino.

ʻO ka mea pōmaikaʻi, hiki iā Hexarelin ke wikiwiki kaumaha lilo ma ka huli ʻana i nā hana kūlohelohe koʻikoʻi i loko o ke kino. Hiki ke kōkua ka hopena wikiwiki o ka momona iā ʻoe i ka hiki ʻana i kāu kaumaha ʻoi aku ka wikiwiki o nā pahu pio ma mua o ka manawa. ʻO ka mea nui, e hana ʻoe pēlā ma kahi palekana a ʻoi aku ka maikaʻi ʻano maikaʻi ke hoʻohālikelike ʻia me nā lāʻau ʻino ʻē aʻe a i ʻole nā ​​papahana ʻai. ʻO ka hui pū ʻana o ka loaʻa ʻana o ka ʻiʻo momona a me ka lean muscle mai Hexarelin hiki ke alakaʻi i kahi hoʻoponopono kino piha.

③ Hoʻomaikaʻi i ka ikaika a me ka maʻalahi

ʻOiai e loaʻa ana i kahi hoʻololi kino holoʻokoʻa, loaʻa iā ʻoe nā pōmaikaʻi o ka hoʻomaikaʻi ʻana i ka ikaika a me ka maʻalahi.

ʻIke ʻia ʻo Hexarelin e hoʻomaikaʻi nui i ka tendon a me ka ikaika ligament. Eia hou, ka pili ka peptide e hoʻonui i ka maʻalahi a me ke olakino hui holoʻokoʻa. He mea koʻikoʻi ka nānā ʻana i nā tendons, ligaments, a me nā ʻiʻo i kou wā ʻelemakule no ka mea e pili ana lākou i ka pōʻino.

No laila, liʻiliʻi ka loaʻa iā ʻoe inā paʻa ʻoe ma ka ʻaoʻao ʻaoʻao ma muli o kahi hōʻeha lōʻihi. ʻAʻole ʻo Hexarelin wale nō e hiki iā ʻoe ke hoʻōla a paʻi koke i ka hale haʻuki akā pale i nā hōʻeha koʻikoʻi ma mua no ka loaʻa ʻana o ka maʻalahi.

④ʻoi aku ka ikaika o ka hoʻihoʻi hou ʻana a me ka hana haʻuki

Loaʻa nā pōmaikaʻi hou i ka lilo ʻana o ke kaumaha, ka loaʻa ʻana o ka ʻiʻo lean, a me ka hoʻomaikaʻi ʻana i ka ikaika holoʻokoʻa.

No ka hoʻomaka, e hoʻōla wikiwiki ʻoe e hāʻawi iā ʻoe i ka manawa e hoʻi ai i ka hale haʻuki a hoʻi i ka hana. Pono ka hoʻihoʻi ʻana kaumaha lilo a me ka loaʻa ʻana o ka ʻiʻo, no laila he mea nui ka loaʻa ʻana o nā mea hoʻohui e kōkua ai i kēlā kaʻina hana.

ʻIke ʻia ʻo Hexarelin e hoʻolalelale wikiwiki mai nā ʻeha a me ke aʻo ʻana. He kū'ē loa ia i nā ʻeha musculoskeletal e hoʻopilikia i ka holomua ma ka hale haʻuki.

Eia kekahi, e ʻike ʻoe i ka holomua holoʻokoʻa o ka hana haʻuki ma muli o ka hopena.

⑤ Hoʻomaikaʻi i ka maikaʻi o ka hiamoe a me ka maikaʻi holoʻokoʻa

ʻO kekahi pōmaikaʻi ʻē aʻe iā Hexarelin nā hōʻike e pili ana i ka hoʻomaikaʻi ʻana o ka peptide i ka maikaʻi o ka hiamoe. ʻO ka hoʻonui ʻana i ka hiki kino me ka hoʻoikaika kuʻuna o ka hoʻoikaika kino e alakaʻi i nā pō maluhia.

A, no ka mea he mea nui ka hiamoe i ke olakino holoʻokoʻa, hāʻawi ka peptide i kahi manaʻo maikaʻi aʻe. ʻO ka lilo ʻana o ke kaumaha a me ka ikaika e alakaʻi i ka hoʻomaikaʻi ʻana iā ʻoe iho a me ka hilinaʻi.

ʻAʻole wale ʻoe e hiamoe maikaʻi akā ʻoi aku ka maikaʻi o ka mahalo i nā hopena maikaʻi o Hexarelin.

Nā hopena ʻaoʻao o Hexarelin

Mahalo, ua hōʻike ʻia aoao waiwai o Hexarelin ka liʻiliʻi.

ʻO ka mea maʻamau aoao waiwai e hoʻokomo i nā manaʻo o ka luhi a i ʻole ka lethargy.[3][4] Ma muli o ka hiki o ka hormone ulu ke hoʻonui i ka makemake no ka hiamoe. Eia naʻe, hiki i ka mālama haʻahaʻa ʻana i ka haʻahaʻa haʻahaʻa hiki ke hoʻopau i kēia pilikia. Hiki ke kōkua i ka hoʻopaʻa ʻana o ka wai i ka ʻoi aku / kiʻekiʻe o Hexarelin.

kekahi hopena ʻaoʻao ʻO ka mea i hōʻike ʻia ʻo ke kani ʻana a i ʻole ka helu ʻana ma nā lima a me nā wāwae.

ʻO ka poʻe i loaʻa nā hōʻailona e hoʻohaʻahaʻa i ka ka hoʻohana ʻana a i ʻole e noʻonoʻo e wehe i ka supplementation pau loa.

ʻOi aku ka maikaʻi e kamaʻilio me ke kauka ma mua o ka hoʻohana ʻana inā ua lawe mua ʻoe i nā lāʻau lapaʻau ʻē aʻe.

Hexarelin me nā peptides ʻē aʻe

Hexarelin vs Ipamorelin

ʻOiai keʻano o ka hana a me ka mea mua pono no nā peptide ʻelua ua like loa, hiki mai ka ʻokoʻa i nā pono lua. Ua hōʻoia ʻia ʻo Ipamorelin e hoʻomaikaʻi i ka nui o ka iwi, aʻo ka hexarelin e hoʻomaikaʻi i ke olakino cardiovascular.

Hexarelin vs GHRP-6

Hana like nā peptides ʻelua. Eia naʻe, ʻaʻole hiki ke hoʻoulu maʻalahi ʻo GHRP-6 (9) i nā ala neuroendocrine ʻē aʻe e like me ka hexarelin. No laila, lanakila ʻo hexarelin i ka heihei kūʻē iā GHRP-6 no ka maopopo!

Ma hea e kūʻai ai i ka Hexarelin?

He hopena koʻikoʻi ka Hexarelin peptide therapy i ke olakino holoʻokoʻa.[1][6] Kōkua ia i ka loaʻa ʻana o ka ʻiʻo, ka metabolizing momona, hoʻonui i ka ikehu, a pēlā aku. Eia ma KANAKA, ua hoʻolaʻa mākou i ka hoʻolako ʻana i nā peptide he nui e pili ana i ka pohō kaumaha, nā mālama olakino olakino, a me nā hormones ʻē aʻe. Inā makemake ʻoe i ka Hexarelin kūʻai nui a i ʻole nā ​​​​peptides ʻē aʻe, e hoʻopiha i ka palapala ma lalo nei e hoʻonohonoho i kāu kūkākūkā a kamaʻilio me kā mākou limahana loea. ʻAʻole hiki iā mākou ke kali i ka lohe ʻana mai iā ʻoe!

Hexarelin Hōʻike Hōʻike-HNMR

He aha ka HNMR a he aha ka HNMR spectrum e haʻi iā ʻoe? ʻO H Nuclear Magnetic Resonance (INMR) spectroscopy kahi ʻenehana kemika analytical i hoʻohana ʻia i ka hoʻokele maikaʻi a me ka noiʻi no ka hoʻoholo ʻana i ka ʻike a me ka maʻemaʻe o kahi laʻana a me kona ʻano molekala. No ka laʻana, hiki i ka NMR ke hoʻokaʻawale i nā hui pū ʻia i ʻike ʻia. No nā pūhui i ʻike ʻole ʻia, hiki ke hoʻohana ʻia ka NMR (a i ʻole e hoʻohālikelike ʻia i nā hale waihona puke spectral a i ʻole e hoʻokaʻawale pololei i ke ʻano kumu. e like me ka hoʻololi conformational, hoʻololi i ka pae, solubility, a me ka diffusion.

Pehea e kūʻai ai iā Hexarelin mai AASraw?

❶I Hoʻokaʻaʻike iā mākou ma kā mākou ʻōnaehana nīnau leka uila, a i ʻole e waiho i kāu helu WhatsApp iā mākou, e hoʻopili aku kā mākou mea kūʻai aku (CSR) iā ʻoe i nā hola 12.

❷E hāʻawi iā mākou i kāu helu a me kāu helu wahi i nīnau ʻia.

❸Na kā mākou CSR e hāʻawi iā ʻoe i ka ʻōlelo ʻōlelo, ka manawa uku, ka helu ʻimi, nā ala lawe, a me ka lā i manaʻo ʻia e hiki mai ai (ETA).

❹E uku ʻia a hoʻouna ʻia nā waiwai i loko o 12 mau hola.

❺ Loaʻa nā waiwai a hāʻawi i nā manaʻo.

Mea kākau o kēia ʻatikala:
Kauka Monique Ua puka 'o Hong mai ke Kula Nui o UK Imperial College London Faculty of Medicine

Mea kākau moʻolelo puke moʻolelo ʻepekema:
1. David Dahlgren
'Oihana o Pharmaceutical Biosciences, Translational Drug Discovery and Development, Uppsala University, Uppsala 752 36, Suedena
2. H. McDonald
Kula o Biomedical Science, University of Queensland, Brisbane, Australia
3. Giuseppe Biagini
Laboratory of Experimental Endocrinology, Department of Internal Medicine, The Sahlgrenska Academy ma ke Kulanui o Gothenburg, Gothenburg, Suedena
4. Anna Barlind
Keʻena o ka Psychiatry, University of Medicine and Dentistry of New Jersey, Robert Wood Johnson Medical School, Piscataway, NJ, USA
ʻAʻole ʻae kēia kauka/ʻepekema i ke kūʻai, kūʻai ʻana, a hoʻohana paha i kēia huahana no kekahi kumu. ʻAʻohe pili a pili ʻole ʻo Aasraw, i hōʻike ʻia a i ʻole, me kēia kauka. ʻO ke kumu o ka haʻi ʻana i kēia kauka, ʻo ia ka hoʻomaikaʻi ʻana a me ka hoʻomaikaʻi ʻana i ka hana noiʻi a me ka hoʻomohala piha i hana ʻia e nā ʻepekema e hana nei i kēia mea.

E hoʻomaopopo '

[1] ʻOmi K (2006). "Hoʻopau i nā lāʻau lapaʻau ma 2005: nā lāʻau lapaʻau cardiovascular". Manaʻo Kuʻuna ma luna o nā lāʻau noiʻi. 15 (11): 1299–308. doi:10.1517/13543784.15.11.1299. PMID 17040192. S2CID 21632578.

[2] Ezio Ghigo (1999). Growth Hormone Secretagogues: Nā ʻike kumu a me nā hopena lapaʻau. Elsevier. aoao 178–. ISBN 978-0-444-82933-7.

[3] Rahim A, O'Neill PA, Shalet SM (1998). "Ke kūlana hormone ulu i ka wā lōʻihi hexarelin therapy". ʻO ka Journal of Clinical Endocrinology & Metabolism. 83 (5): 1644–9. doi:10.1210/jcem.83.5.4812. PMID 9589671.

[4] Ghigo E, Arvat E, Gianotti L, Imbimbo BP, Lenaerts V, Deghenghi R, et al. (1994). "Ka hana hoʻokuʻu ʻana i ka hormone ulu o hexarelin, he hexapeptide synthetic hou, ma hope o ka intravenous, subcutaneous, intranasal, a me ka hoʻokele waha i ke kanaka". ʻO ka Journal of Clinical Endocrinology & Metabolism. 78 (3): 693–8. doi:10.1210/jcem.78.3.8126144. PMID 8126144.

[5] Imbimbo, BP; Mant, T.; Edwards, M.; Amin, D.; Dalton, N.; Boutignon, F.; Lenaerts, V.; Wďż˝thrich, P.; Deghenghi, R. (1994). "Ka hana hoʻokuʻu ʻana i ka hormone ulu o ka hexarelin i nā kānaka". European Journal of Clinical Pharmacology. 46 (5): 421–5. doi:10.1007/bf00191904. PMID 7957536. S2CID 19573322.

[6] CR Ganellin; ʻO David J. Triggle (21 Nowemapa 1996). ʻO ka puke wehewehe ʻōlelo o nā Agena Pharmacological. CRC Press. aoao 617–. ISBN 978-0-412-46630-4.


E kiʻi i kahi hōʻaiʻē nui